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8PKW

Kelch domain of KEAP1 in complex with a ortho-dimethylbenzene linked cyclic peptide 5 (ortho-WRCDPETaEC).

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSITE: Sensor for electrophilic agents => ECO:0000250|UniProtKB:Q9Z2X8
ChainResidueDetails
ACYS434
BCYS434

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: S-(2-succinyl)cysteine => ECO:0000250|UniProtKB:Q9Z2X8
ChainResidueDetails
ASER319
ASER613
BSER319
BSER613

site_idSWS_FT_FI3
Number of Residues2
DetailsMOD_RES: S-cGMP-cysteine => ECO:0000250|UniProtKB:Q9Z2X8
ChainResidueDetails
ACYS434
BCYS434

219869

PDB entries from 2024-05-15

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