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8GPR

GluK1-1a receptor captured in the desensitized state

Functional Information from GO Data
ChainGOidnamespacecontents
A0000149molecular_functionSNARE binding
A0004970molecular_functionglutamate-gated receptor activity
A0005216molecular_functionmonoatomic ion channel activity
A0005234molecular_functionextracellularly glutamate-gated ion channel activity
A0005313molecular_functionL-glutamate transmembrane transporter activity
A0005515molecular_functionprotein binding
A0005886cellular_componentplasma membrane
A0006811biological_processmonoatomic ion transport
A0007215biological_processglutamate receptor signaling pathway
A0007268biological_processchemical synaptic transmission
A0007399biological_processnervous system development
A0008328cellular_componentionotropic glutamate receptor complex
A0014054biological_processpositive regulation of gamma-aminobutyric acid secretion
A0014069cellular_componentpostsynaptic density
A0015276molecular_functionligand-gated monoatomic ion channel activity
A0015277molecular_functionkainate selective glutamate receptor activity
A0015813biological_processL-glutamate transmembrane transport
A0016020cellular_componentmembrane
A0016595molecular_functionglutamate binding
A0019722biological_processcalcium-mediated signaling
A0022849molecular_functionglutamate-gated calcium ion channel activity
A0030425cellular_componentdendrite
A0030534biological_processadult behavior
A0032229biological_processnegative regulation of synaptic transmission, GABAergic
A0032230biological_processpositive regulation of synaptic transmission, GABAergic
A0032983cellular_componentkainate selective glutamate receptor complex
A0034220biological_processmonoatomic ion transmembrane transport
A0035235biological_processionotropic glutamate receptor signaling pathway
A0035249biological_processsynaptic transmission, glutamatergic
A0038023molecular_functionsignaling receptor activity
A0042391biological_processregulation of membrane potential
A0042734cellular_componentpresynaptic membrane
A0042802molecular_functionidentical protein binding
A0043025cellular_componentneuronal cell body
A0043195cellular_componentterminal bouton
A0043235cellular_componentreceptor complex
A0045202cellular_componentsynapse
A0045211cellular_componentpostsynaptic membrane
A0048167biological_processregulation of synaptic plasticity
A0048172biological_processregulation of short-term neuronal synaptic plasticity
A0048266biological_processbehavioral response to pain
A0050804biological_processmodulation of chemical synaptic transmission
A0051899biological_processmembrane depolarization
A0051967biological_processnegative regulation of synaptic transmission, glutamatergic
A0060079biological_processexcitatory postsynaptic potential
A0060080biological_processinhibitory postsynaptic potential
A0097110molecular_functionscaffold protein binding
A0098815biological_processmodulation of excitatory postsynaptic potential
A0098839cellular_componentpostsynaptic density membrane
A0098978cellular_componentglutamatergic synapse
A0099505biological_processregulation of presynaptic membrane potential
A0099507molecular_functionligand-gated monoatomic ion channel activity involved in regulation of presynaptic membrane potential
A1901363molecular_functionheterocyclic compound binding
A1904315molecular_functiontransmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential
B0000149molecular_functionSNARE binding
B0004970molecular_functionglutamate-gated receptor activity
B0005216molecular_functionmonoatomic ion channel activity
B0005234molecular_functionextracellularly glutamate-gated ion channel activity
B0005313molecular_functionL-glutamate transmembrane transporter activity
B0005515molecular_functionprotein binding
B0005886cellular_componentplasma membrane
B0006811biological_processmonoatomic ion transport
B0007215biological_processglutamate receptor signaling pathway
B0007268biological_processchemical synaptic transmission
B0007399biological_processnervous system development
B0008328cellular_componentionotropic glutamate receptor complex
B0014054biological_processpositive regulation of gamma-aminobutyric acid secretion
B0014069cellular_componentpostsynaptic density
B0015276molecular_functionligand-gated monoatomic ion channel activity
B0015277molecular_functionkainate selective glutamate receptor activity
B0015813biological_processL-glutamate transmembrane transport
B0016020cellular_componentmembrane
B0016595molecular_functionglutamate binding
B0019722biological_processcalcium-mediated signaling
B0022849molecular_functionglutamate-gated calcium ion channel activity
B0030425cellular_componentdendrite
B0030534biological_processadult behavior
B0032229biological_processnegative regulation of synaptic transmission, GABAergic
B0032230biological_processpositive regulation of synaptic transmission, GABAergic
B0032983cellular_componentkainate selective glutamate receptor complex
B0034220biological_processmonoatomic ion transmembrane transport
B0035235biological_processionotropic glutamate receptor signaling pathway
B0035249biological_processsynaptic transmission, glutamatergic
B0038023molecular_functionsignaling receptor activity
B0042391biological_processregulation of membrane potential
B0042734cellular_componentpresynaptic membrane
B0042802molecular_functionidentical protein binding
B0043025cellular_componentneuronal cell body
B0043195cellular_componentterminal bouton
B0043235cellular_componentreceptor complex
B0045202cellular_componentsynapse
B0045211cellular_componentpostsynaptic membrane
B0048167biological_processregulation of synaptic plasticity
B0048172biological_processregulation of short-term neuronal synaptic plasticity
B0048266biological_processbehavioral response to pain
B0050804biological_processmodulation of chemical synaptic transmission
B0051899biological_processmembrane depolarization
B0051967biological_processnegative regulation of synaptic transmission, glutamatergic
B0060079biological_processexcitatory postsynaptic potential
B0060080biological_processinhibitory postsynaptic potential
B0097110molecular_functionscaffold protein binding
B0098815biological_processmodulation of excitatory postsynaptic potential
B0098839cellular_componentpostsynaptic density membrane
B0098978cellular_componentglutamatergic synapse
B0099505biological_processregulation of presynaptic membrane potential
B0099507molecular_functionligand-gated monoatomic ion channel activity involved in regulation of presynaptic membrane potential
B1901363molecular_functionheterocyclic compound binding
B1904315molecular_functiontransmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential
C0000149molecular_functionSNARE binding
C0004970molecular_functionglutamate-gated receptor activity
C0005216molecular_functionmonoatomic ion channel activity
C0005234molecular_functionextracellularly glutamate-gated ion channel activity
C0005313molecular_functionL-glutamate transmembrane transporter activity
C0005515molecular_functionprotein binding
C0005886cellular_componentplasma membrane
C0006811biological_processmonoatomic ion transport
C0007215biological_processglutamate receptor signaling pathway
C0007268biological_processchemical synaptic transmission
C0007399biological_processnervous system development
C0008328cellular_componentionotropic glutamate receptor complex
C0014054biological_processpositive regulation of gamma-aminobutyric acid secretion
C0014069cellular_componentpostsynaptic density
C0015276molecular_functionligand-gated monoatomic ion channel activity
C0015277molecular_functionkainate selective glutamate receptor activity
C0015813biological_processL-glutamate transmembrane transport
C0016020cellular_componentmembrane
C0016595molecular_functionglutamate binding
C0019722biological_processcalcium-mediated signaling
C0022849molecular_functionglutamate-gated calcium ion channel activity
C0030425cellular_componentdendrite
C0030534biological_processadult behavior
C0032229biological_processnegative regulation of synaptic transmission, GABAergic
C0032230biological_processpositive regulation of synaptic transmission, GABAergic
C0032983cellular_componentkainate selective glutamate receptor complex
C0034220biological_processmonoatomic ion transmembrane transport
C0035235biological_processionotropic glutamate receptor signaling pathway
C0035249biological_processsynaptic transmission, glutamatergic
C0038023molecular_functionsignaling receptor activity
C0042391biological_processregulation of membrane potential
C0042734cellular_componentpresynaptic membrane
C0042802molecular_functionidentical protein binding
C0043025cellular_componentneuronal cell body
C0043195cellular_componentterminal bouton
C0043235cellular_componentreceptor complex
C0045202cellular_componentsynapse
C0045211cellular_componentpostsynaptic membrane
C0048167biological_processregulation of synaptic plasticity
C0048172biological_processregulation of short-term neuronal synaptic plasticity
C0048266biological_processbehavioral response to pain
C0050804biological_processmodulation of chemical synaptic transmission
C0051899biological_processmembrane depolarization
C0051967biological_processnegative regulation of synaptic transmission, glutamatergic
C0060079biological_processexcitatory postsynaptic potential
C0060080biological_processinhibitory postsynaptic potential
C0097110molecular_functionscaffold protein binding
C0098815biological_processmodulation of excitatory postsynaptic potential
C0098839cellular_componentpostsynaptic density membrane
C0098978cellular_componentglutamatergic synapse
C0099505biological_processregulation of presynaptic membrane potential
C0099507molecular_functionligand-gated monoatomic ion channel activity involved in regulation of presynaptic membrane potential
C1901363molecular_functionheterocyclic compound binding
C1904315molecular_functiontransmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential
D0000149molecular_functionSNARE binding
D0004970molecular_functionglutamate-gated receptor activity
D0005216molecular_functionmonoatomic ion channel activity
D0005234molecular_functionextracellularly glutamate-gated ion channel activity
D0005313molecular_functionL-glutamate transmembrane transporter activity
D0005515molecular_functionprotein binding
D0005886cellular_componentplasma membrane
D0006811biological_processmonoatomic ion transport
D0007215biological_processglutamate receptor signaling pathway
D0007268biological_processchemical synaptic transmission
D0007399biological_processnervous system development
D0008328cellular_componentionotropic glutamate receptor complex
D0014054biological_processpositive regulation of gamma-aminobutyric acid secretion
D0014069cellular_componentpostsynaptic density
D0015276molecular_functionligand-gated monoatomic ion channel activity
D0015277molecular_functionkainate selective glutamate receptor activity
D0015813biological_processL-glutamate transmembrane transport
D0016020cellular_componentmembrane
D0016595molecular_functionglutamate binding
D0019722biological_processcalcium-mediated signaling
D0022849molecular_functionglutamate-gated calcium ion channel activity
D0030425cellular_componentdendrite
D0030534biological_processadult behavior
D0032229biological_processnegative regulation of synaptic transmission, GABAergic
D0032230biological_processpositive regulation of synaptic transmission, GABAergic
D0032983cellular_componentkainate selective glutamate receptor complex
D0034220biological_processmonoatomic ion transmembrane transport
D0035235biological_processionotropic glutamate receptor signaling pathway
D0035249biological_processsynaptic transmission, glutamatergic
D0038023molecular_functionsignaling receptor activity
D0042391biological_processregulation of membrane potential
D0042734cellular_componentpresynaptic membrane
D0042802molecular_functionidentical protein binding
D0043025cellular_componentneuronal cell body
D0043195cellular_componentterminal bouton
D0043235cellular_componentreceptor complex
D0045202cellular_componentsynapse
D0045211cellular_componentpostsynaptic membrane
D0048167biological_processregulation of synaptic plasticity
D0048172biological_processregulation of short-term neuronal synaptic plasticity
D0048266biological_processbehavioral response to pain
D0050804biological_processmodulation of chemical synaptic transmission
D0051899biological_processmembrane depolarization
D0051967biological_processnegative regulation of synaptic transmission, glutamatergic
D0060079biological_processexcitatory postsynaptic potential
D0060080biological_processinhibitory postsynaptic potential
D0097110molecular_functionscaffold protein binding
D0098815biological_processmodulation of excitatory postsynaptic potential
D0098839cellular_componentpostsynaptic density membrane
D0098978cellular_componentglutamatergic synapse
D0099505biological_processregulation of presynaptic membrane potential
D0099507molecular_functionligand-gated monoatomic ion channel activity involved in regulation of presynaptic membrane potential
D1901363molecular_functionheterocyclic compound binding
D1904315molecular_functiontransmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI2
Number of Residues16
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"15710405","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1YCJ","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues8
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"15710405","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"15721240","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1YCJ","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues160
DetailsTransmembrane: {"description":"Helical","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues4
DetailsModified residue: {"description":"Phosphoserine; by PKC","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues4
DetailsModified residue: {"description":"Phosphothreonine; by PKC","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues32
DetailsGlycosylation: {"description":"N-linked (GlcNAc...) asparagine","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

246333

PDB entries from 2025-12-17

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