8E0G
Re-refined model of active mu-opioid receptor (PDB 5c1m) as an adduct with BU72
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0004930 | molecular_function | G protein-coupled receptor activity |
A | 0004979 | molecular_function | beta-endorphin receptor activity |
A | 0004985 | molecular_function | G protein-coupled opioid receptor activity |
A | 0007186 | biological_process | G protein-coupled receptor signaling pathway |
A | 0016020 | cellular_component | membrane |
Functional Information from PROSITE/UniProt
site_id | PS00237 |
Number of Residues | 17 |
Details | G_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. TSIfTLCTMSVDRYIaV |
Chain | Residue | Details |
A | THR153-VAL169 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 24 |
Details | TRANSMEM: Helical; Name=1 => ECO:0000269|PubMed:22437502, ECO:0000269|PubMed:26245379 |
Chain | Residue | Details |
A | THR67-TYR91 |
site_id | SWS_FT_FI2 |
Number of Residues | 54 |
Details | TOPO_DOM: Cytoplasmic => ECO:0000269|PubMed:22437502, ECO:0000269|PubMed:26245379 |
Chain | Residue | Details |
A | VAL92-ASN104 | |
A | ASP164-ASN183 | |
A | LEU254-ARG277 |
site_id | SWS_FT_FI3 |
Number of Residues | 24 |
Details | TRANSMEM: Helical; Name=2 => ECO:0000269|PubMed:22437502, ECO:0000269|PubMed:26245379 |
Chain | Residue | Details |
A | ILE105-LEU129 |
site_id | SWS_FT_FI4 |
Number of Residues | 39 |
Details | TOPO_DOM: Extracellular => ECO:0000269|PubMed:22437502, ECO:0000269|PubMed:26245379 |
Chain | Residue | Details |
A | MET130-CYS140 | |
A | ALA206-TRP228 | |
A | LEU305-THR312 |
site_id | SWS_FT_FI5 |
Number of Residues | 22 |
Details | TRANSMEM: Helical; Name=3 => ECO:0000269|PubMed:22437502, ECO:0000269|PubMed:26245379 |
Chain | Residue | Details |
A | LYS141-VAL163 |
site_id | SWS_FT_FI6 |
Number of Residues | 21 |
Details | TRANSMEM: Helical; Name=4 => ECO:0000269|PubMed:22437502, ECO:0000269|PubMed:26245379 |
Chain | Residue | Details |
A | ALA184-MET205 |
site_id | SWS_FT_FI7 |
Number of Residues | 24 |
Details | TRANSMEM: Helical; Name=5 => ECO:0000269|PubMed:22437502, ECO:0000269|PubMed:26245379 |
Chain | Residue | Details |
A | GLU229-GLY253 |
site_id | SWS_FT_FI8 |
Number of Residues | 26 |
Details | TRANSMEM: Helical; Name=6 => ECO:0000269|PubMed:22437502, ECO:0000269|PubMed:26245379 |
Chain | Residue | Details |
A | ILE278-ALA304 |
site_id | SWS_FT_FI9 |
Number of Residues | 23 |
Details | TRANSMEM: Helical; Name=7 => ECO:0000269|PubMed:22437502, ECO:0000269|PubMed:26245379 |
Chain | Residue | Details |
A | PHE313-TYR336 |
site_id | SWS_FT_FI10 |
Number of Residues | 1 |
Details | MOD_RES: Phosphotyrosine => ECO:0000250|UniProtKB:P33535 |
Chain | Residue | Details |
A | TYR166 |