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7W3P

Crystal structure of RORgamma in complex with natural inverse agonist

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsMotif: {"description":"AF-2"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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