7TRB
CRYSTAL STRUCTURE OF FARNESOID X-ACTIVATED RECEPTOR COMPLEXED WITH COMPOUND-32 AKA (1S,3S)-N-({4-[5-(2-FLUOROPR OPAN-2-YL)-1,2,4-OXADIAZOL-3-YL]BICYCLO[2.2.2]OCTAN-1-YL}M ETHYL)-3-HYDROXY-N-[4'-(2-HYDROXYPROPAN-2-YL)-[1,1'-BIPHEN YL]-3-YL]-3-(TRIFLUOROMETHYL)CYCLOBUTANE-1-CARBOXAMIDE
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0003677 | molecular_function | DNA binding |
A | 0004879 | molecular_function | nuclear receptor activity |
A | 0006355 | biological_process | regulation of DNA-templated transcription |
A | 0032052 | molecular_function | bile acid binding |
A | 0038183 | biological_process | bile acid signaling pathway |
B | 0003677 | molecular_function | DNA binding |
B | 0004879 | molecular_function | nuclear receptor activity |
B | 0006355 | biological_process | regulation of DNA-templated transcription |
B | 0032052 | molecular_function | bile acid binding |
B | 0038183 | biological_process | bile acid signaling pathway |
Functional Information from SwissProt/UniProt
Chain | Residue | Details |
A | ARG335 | |
A | TYR365 | |
A | TYR373 | |
A | HIS451 | |
B | ARG335 | |
B | TYR365 | |
B | TYR373 | |
B | HIS451 | |
Chain | Residue | Details |
A | THR446 | |
B | THR446 | |
site_id | SWS_FT_FI3 |
Number of Residues | 4 |
Details | CROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO1) => ECO:0000305|PubMed:23546875 |
Chain | Residue | Details |
A | LYS279 | |
B | LYS279 | |