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7OR4

Crystal structure of DPP8 in complex with a 4-oxo-b-lactam based inhibitor, B142

Functional Information from GO Data
ChainGOidnamespacecontents
A0004177molecular_functionaminopeptidase activity
A0005515molecular_functionprotein binding
A0005737cellular_componentcytoplasm
A0005829cellular_componentcytosol
A0006508biological_processproteolysis
A0006915biological_processapoptotic process
A0006955biological_processimmune response
A0008233molecular_functionpeptidase activity
A0008236molecular_functionserine-type peptidase activity
A0008239molecular_functiondipeptidyl-peptidase activity
A0016787molecular_functionhydrolase activity
A0043069biological_processnegative regulation of programmed cell death
A0051604biological_processprotein maturation
A0140633biological_processCARD8 inflammasome complex assembly
A0141201biological_processpyroptotic cell death
A1904784biological_processNLRP1 inflammasome complex assembly
B0004177molecular_functionaminopeptidase activity
B0005515molecular_functionprotein binding
B0005737cellular_componentcytoplasm
B0005829cellular_componentcytosol
B0006508biological_processproteolysis
B0006915biological_processapoptotic process
B0006955biological_processimmune response
B0008233molecular_functionpeptidase activity
B0008236molecular_functionserine-type peptidase activity
B0008239molecular_functiondipeptidyl-peptidase activity
B0016787molecular_functionhydrolase activity
B0043069biological_processnegative regulation of programmed cell death
B0051604biological_processprotein maturation
B0140633biological_processCARD8 inflammasome complex assembly
B0141201biological_processpyroptotic cell death
B1904784biological_processNLRP1 inflammasome complex assembly
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsACT_SITE: Charge relay system => ECO:0000305|PubMed:12534281, ECO:0000305|PubMed:29382749
ChainResidueDetails
BSER755
BASP833
BHIS865
ASER755
AASP833
AHIS865

238268

PDB entries from 2025-07-02

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