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7OF9

Keap1 kelch domain bound to a small molecule fragment

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue VBK A 701
ChainResidue
ATYR334
AARG415
ASER555
AALA556

site_idAC2
Number of Residues5
Detailsbinding site for residue DMS A 702
ChainResidue
AARG354
ALEU355
AASP357
AHIS552
ALEU578

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Sensor for electrophilic agents => ECO:0000269|PubMed:20498371
ChainResidueDetails
ACYS434

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: S-cGMP-cysteine => ECO:0000269|PubMed:20498371
ChainResidueDetails
ACYS434

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: S-(2-succinyl)cysteine => ECO:0000269|PubMed:22014577
ChainResidueDetails
ACYS613

222415

PDB entries from 2024-07-10

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