7OE9
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH rac-N5-((1R,5S)-3-oxabicyclo[3.1.0]hexan-6-yl)-N7,3-dimethyl-3-phenyl-2,3-dihydrobenzofuran-5,7-dicarboxamide
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 11 |
Details | binding site for residue V9N A 501 |
Chain | Residue |
A | LYS351 |
A | HOH644 |
A | HOH688 |
A | TRP370 |
A | PRO371 |
A | LEU383 |
A | TYR428 |
A | ASN429 |
A | PRO430 |
A | MET438 |
A | HOH621 |
site_id | AC2 |
Number of Residues | 6 |
Details | binding site for residue EDO A 502 |
Chain | Residue |
A | TYR426 |
A | ARG440 |
A | GLN443 |
A | GLN443 |
A | ASP444 |
A | HOH601 |
site_id | AC3 |
Number of Residues | 5 |
Details | binding site for residue EDO A 503 |
Chain | Residue |
A | LYS402 |
A | ASP407 |
A | MET438 |
A | LYS441 |
A | HOH602 |
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 60 |
Details | BROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY |
Chain | Residue | Details |
A | ALA369-TYR428 | |