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7NQJ

C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH N-ethyl-2-(1-methyl-1H-1,2,3-triazol-4-yl)-6-(1-phenylethyl)isonicotinamide

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue UME A 501
ChainResidue
APRO371
AVAL376
ALEU383
ATYR428
AASN429
AHIS433
AVAL435
AHOH615
AHOH665

site_idAC2
Number of Residues7
Detailsbinding site for residue EDO A 502
ChainResidue
ATYR426
AARG440
AGLN443
AGLN443
AASP444
APHE448
AHOH601

site_idAC3
Number of Residues5
Detailsbinding site for residue EDO A 503
ChainResidue
ALYS402
AASP407
AMET438
ALYS441
AHOH602

site_idAC4
Number of Residues4
Detailsbinding site for residue EDO A 504
ChainResidue
ALYS427
ATYR428
AASN429
AHOH669

site_idAC5
Number of Residues3
Detailsbinding site for residue PEG A 505
ChainResidue
ASER347
ALYS351
AHOH668

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

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PDB entries from 2024-10-16

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