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7MSA

GDC-9545 in complex with estrogen receptor alpha

Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue G9J D 601
ChainResidue
DLEU346
DLEU525
DHOH705
DTHR347
DALA350
DGLU353
DLEU387
DARG394
DILE424
DGLY521
DHIS524

site_idAC2
Number of Residues15
Detailsbinding site for residue ZNM A 601
ChainResidue
AMET343
ALEU346
ATHR347
AASP351
AGLU353
ALEU354
ATRP383
ALEU384
AARG394
APHE404
AMET421
AILE424
AGLY521
AHIS524
ALEU525

site_idAC3
Number of Residues14
Detailsbinding site for residue ZNM C 601
ChainResidue
CMET343
CLEU346
CTHR347
CASP351
CGLU353
CLEU384
CLEU387
CMET388
CARG394
CMET421
CGLY521
CHIS524
CLEU525
CPRO535

site_idAC4
Number of Residues10
Detailsbinding site for residue G9J B 601
ChainResidue
BLEU346
BTHR347
BALA350
BGLU353
BLEU387
BARG394
BILE424
BGLY521
BHIS524
BLEU525

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ATYR537
CTYR537
BTYR537
DTYR537

site_idSWS_FT_FI2
Number of Residues4
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447
CCYS447
BCYS447
DCYS447

220472

PDB entries from 2024-05-29

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