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7LB2

Crystal structure of the tandem bromodomain (BD1, BD2) of human TAF1 bound to ZS1-589

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0005669cellular_componenttranscription factor TFIID complex
A0006366biological_processtranscription by RNA polymerase II
A0016251molecular_functionRNA polymerase II general transcription initiation factor activity
A0017025molecular_functionTBP-class protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue EDO A 1801
ChainResidue
AARG1397
AHIS1406
AGLN1428
AARG1431

site_idAC2
Number of Residues5
Detailsbinding site for residue EDO A 1802
ChainResidue
APHE1405
AASN1460
AEDO1807
AEDO1808
AHOH1919

site_idAC3
Number of Residues5
Detailsbinding site for residue EDO A 1803
ChainResidue
AMET1520
AASP1524
ASER1525
ATRP1526
AHOH1901

site_idAC4
Number of Residues3
Detailsbinding site for residue EDO A 1804
ChainResidue
ATRP1526
AHIS1529
AHOH1942

site_idAC5
Number of Residues4
Detailsbinding site for residue HEZ A 1805
ChainResidue
AASN1546
ALYS1561
ASER1567
AASP1570

site_idAC6
Number of Residues2
Detailsbinding site for residue EDO A 1806
ChainResidue
AHOH1937
AHOH1945

site_idAC7
Number of Residues5
Detailsbinding site for residue EDO A 1807
ChainResidue
ATYR1459
AASN1460
ALEU1466
AEDO1802
AHOH1972

site_idAC8
Number of Residues9
Detailsbinding site for residue EDO A 1808
ChainResidue
APRO1404
ATHR1407
APRO1408
AVAL1409
AASN1410
AEDO1802
AHOH1922
AHOH1972
AHOH2023

site_idAC9
Number of Residues5
Detailsbinding site for residue EDO A 1809
ChainResidue
ASER1441
AGLU1444
ALEU1499
ALYS1559
AHOH1981

site_idAD1
Number of Residues9
Detailsbinding site for residue XWY A 1810
ChainResidue
ATRP1526
APRO1527
AHIS1530
APRO1531
AVAL1532
AASN1533
APHE1536
AASN1583
ATYR1589

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. TypFhtpvNakvvk..DYYkiItrpMdlqtLrenvrkrl..Ypsreefrehlel.IvkNSatY
ChainResidueDetails
ATHR1402-TYR1459
ASER1525-TYR1582

222415

PDB entries from 2024-07-10

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