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7L9G

Crystal structure of the second bromodomain (BD2) of human BRD2 bound to BI2536

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 501
ChainResidue
AHIS433
AASP434
AMET438
AR78503
AHOH604
AHOH648

site_idAC2
Number of Residues2
Detailsbinding site for residue EDO A 502
ChainResidue
ALEU346
AARG406

site_idAC3
Number of Residues9
Detailsbinding site for residue R78 A 503
ChainResidue
AVAL376
ALEU383
ACYS425
AASN429
AHIS433
AEDO501
AHOH629
AHOH710
APRO371

site_idAC4
Number of Residues4
Detailsbinding site for residue CL A 504
ChainResidue
AARG419
AARG419
AHOH661
AHOH661

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

221051

PDB entries from 2024-06-12

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