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7L6D

Crystal structure of the second bromodomain (BD2) of human BRD2 bound to bromosporine

Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue BMF A 501
ChainResidue
ATRP370
AEDO506
AEDO507
AHOH612
AHOH642
AHOH651
APRO371
ALYS374
APRO375
AVAL376
AASP377
ALEU381
AASN429
AEDO504

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 502
ChainResidue
ATRP370
AHIS433
AEDO504
AHOH643

site_idAC3
Number of Residues7
Detailsbinding site for residue EDO A 503
ChainResidue
AILE389
AILE390
ALYS391
AHIS392
AASN424
ALYS427
AASP455

site_idAC4
Number of Residues7
Detailsbinding site for residue EDO A 504
ChainResidue
APRO375
ATHR398
AARG401
ABMF501
AEDO502
AEDO506
AHOH618

site_idAC5
Number of Residues5
Detailsbinding site for residue EDO A 505
ChainResidue
AHIS387
AILE390
ALYS391
APRO393
AHOH641

site_idAC6
Number of Residues7
Detailsbinding site for residue EDO A 506
ChainResidue
ALEU381
APRO393
ATHR398
ABMF501
AEDO504
AHOH625
AHOH643

site_idAC7
Number of Residues5
Detailsbinding site for residue EDO A 507
ChainResidue
AASP377
AHIS392
ABMF501
AHOH616
AHOH638

site_idAC8
Number of Residues5
Detailsbinding site for residue EDO A 508
ChainResidue
ASER362
ALYS363
ALYS363
ALYS364
AHOH653

site_idAC9
Number of Residues3
Detailsbinding site for residue EDO A 509
ChainResidue
AASP388
AHOH641
AHOH680

site_idAD1
Number of Residues6
Detailsbinding site for residue SO4 A 510
ChainResidue
AASN354
AASN354
AGLU404
AARG406
AARG406
AHOH603

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

237735

PDB entries from 2025-06-18

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