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7K7Q

CRYSTAL STRUCTURE OF TYROSINE KINASE 2 JH2 (PSEUDO KINASE DOMAIN) COMPLEXED WITH COMPOUND-12 AKA:6-[(cyclopropanecarbonyl)amino]-4-({3-[6-(dimethylcarbamoyl)pyridazin-3-yl]-2-methoxyphenyl}amino)-N-methylpyridazine-3-carboxamide

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues19
Detailsbinding site for residue VZG A 901
ChainResidue
AGLN597
AVAL690
AGLU691
AHIS692
AGLY693
ACYS736
AARG738
AASN739
ALEU741
ASER758
AHOH1026
AGLY598
ATHR599
AVAL640
ALYS642
AALA671
ATHR687
AGLU688
ATYR689

site_idAC2
Number of Residues19
Detailsbinding site for residue VZG B 901
ChainResidue
BGLN597
BGLY598
BTHR599
BVAL640
BLYS642
BALA671
BTHR687
BGLU688
BVAL690
BGLU691
BGLY693
BASN734
BCYS736
BARG738
BASN739
BLEU741
BSER758
BARG775
BHOH1009

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphotyrosine => ECO:0000250|UniProtKB:Q9R117
ChainResidueDetails
BTYR604
ATYR604

219869

PDB entries from 2024-05-15

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