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7K27

Crystal structure of the tandem bromodomain (BD1, BD2) of human TAF1 bound to ATR inhibitor AZ20

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0005669cellular_componenttranscription factor TFIID complex
A0006366biological_processtranscription by RNA polymerase II
A0016251molecular_functionRNA polymerase II general transcription initiation factor activity
A0017025molecular_functionTBP-class protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue EDO A 1701
ChainResidue
APHE1405
AASN1460
ALEU1466
AHOH1845
AHOH1851
AHOH1853
AHOH1909

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 1702
ChainResidue
ASER1525
ATRP1526
AMET1520
AASP1524

site_idAC3
Number of Residues4
Detailsbinding site for residue EDO A 1703
ChainResidue
AVAL1532
AHOH1878
AHOH1933
AHOH1981

site_idAC4
Number of Residues4
Detailsbinding site for residue EDO A 1704
ChainResidue
ATHR1407
APRO1408
AASN1410
AHOH1803

site_idAC5
Number of Residues10
Detailsbinding site for residue VCD A 1705
ChainResidue
ATRP1526
APRO1527
APHE1528
AHIS1530
APRO1531
AASN1533
ATYR1582
AASN1583
ATYR1589
AHOH1920

site_idAC6
Number of Residues2
Detailsbinding site for residue DMS A 1706
ChainResidue
AASP1539
ATYR1582

site_idAC7
Number of Residues5
Detailsbinding site for residue GOL A 1707
ChainResidue
ALYS1561
ASER1567
AASP1570
AASP1571
AHOH1805

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. TypFhtpvNakvvk..DYYkiItrpMdlqtLrenvrkrl..Ypsreefrehlel.IvkNSatY
ChainResidueDetails
ATHR1402-TYR1459
ASER1525-TYR1582

224931

PDB entries from 2024-09-11

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