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7K03

Crystal structure of the tandem bromodomain (BD1 and BD2) of human TAF1 bound to ATR kinase inhibitor AZD6738

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0005669cellular_componenttranscription factor TFIID complex
A0006366biological_processtranscription by RNA polymerase II
A0016251molecular_functionRNA polymerase II general transcription initiation factor activity
A0017025molecular_functionTBP-class protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue VJM A 1701
ChainResidue
ATRP1526
AHOH1945
AHOH1967
AHOH1975
AHOH2005
APRO1527
APHE1528
AHIS1530
APRO1531
AVAL1532
AASN1533
AASN1583
ATYR1589

site_idAC2
Number of Residues6
Detailsbinding site for residue EDO A 1702
ChainResidue
APRO1404
AASN1460
AHOH1826
AHOH1845
AHOH1852
AHOH2029

site_idAC3
Number of Residues3
Detailsbinding site for residue EDO A 1703
ChainResidue
AARG1423
APRO1424
AMET1425

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 1704
ChainResidue
ALYS1561
ASER1567
AASP1570
AASP1571
AHOH1810

site_idAC5
Number of Residues8
Detailsbinding site for residue EDO A 1705
ChainResidue
AMET1520
AVAL1522
AASP1524
ASER1525
ATRP1526
AHIS1529
AHOH1801
AHOH1899

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. TypFhtpvNakvvk..DYYkiItrpMdlqtLrenvrkrl..Ypsreefrehlel.IvkNSatY
ChainResidueDetails
ATHR1402-TYR1459
ASER1525-TYR1582

221051

PDB entries from 2024-06-12

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