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7JYM

CRYSTAL STRUCTURE OF RAR-RELATED ORPHAN RECEPTOR C (NHIS-RORGT(244-487)-L6-SRC1(678-692)) IN COMPLEX WITH A TRICYCLIC SULFONE INVERSE AGONIST

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues18
Detailsbinding site for residue Z8I A 4000
ChainResidue
AGLN286
APHE377
APHE378
APHE388
ALEU391
ALEU396
AILE397
AILE400
APHE401
AHIS479
ALEU287
ACYS320
AHIS323
ALEU324
AALA327
AARG364
AMET365
AALA368

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsMotif: {"description":"AF-2"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 4"}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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