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7JTM

CRYSTAL STRUCTURE OF RAR-RELATED ORPHAN RECEPTOR C (NHIS-RORGT(244-487)-L6-SRC1(6T78-692) IN COMPLEX WITH A TRICYCLIC SULFONE RORGT INVERSE AGONIST

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues20
Detailsbinding site for residue VK7 A 4000
ChainResidue
AGLN286
AARG367
APHE378
APHE388
ALEU391
ALEU396
AILE397
AILE400
APHE401
AHIS479
AHOH4103
ALEU287
AHOH4106
ACYS320
AALA321
AHIS323
ALEU324
AMET358
AARG364
AMET365

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsMotif: {"description":"AF-2"}
ChainResidueDetails

249697

PDB entries from 2026-02-25

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