Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

7JSP

Crystal structure of the second bromodomain (BD2) of human TAF1 bound to ATR kinase inhibitor AZD6738

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0005669cellular_componenttranscription factor TFIID complex
A0006366biological_processtranscription by RNA polymerase II
A0016251molecular_functionRNA polymerase II general transcription initiation factor activity
A0017025molecular_functionTBP-class protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue VJM A 1701
ChainResidue
ATRP1526
ATYR1589
ATYR1601
AEDO1702
AHOH1882
APRO1527
AHIS1530
APRO1531
AVAL1532
AASN1533
APHE1536
ALEU1569
AASN1583

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 1702
ChainResidue
AARG1565
AVJM1701
AHOH1818
AHOH1821

site_idAC3
Number of Residues4
Detailsbinding site for residue SO4 A 1703
ChainResidue
ALYS1581
ATYR1582
AASN1583
AGLY1584

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. SwpFhhpvNkkfvp..DYYkvIvnpMdletIrkniskhk..Yqsresflddvnl.IlaNSvkY
ChainResidueDetails
ASER1525-TYR1582

221051

PDB entries from 2024-06-12

PDB statisticsPDBj update infoContact PDBjnumon