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7JKX

Bromodomain-containing protein 4 (BRD4) bromodomain 1 (BD1) complexed with YF3-6

Functional Information from PDB Data
site_idAC1
Number of Residues18
Detailsbinding site for residue Y36 A 201
ChainResidue
APRO53
ALEU92
ALEU94
ATYR139
AASN140
AASP145
AMET149
AHOH309
AHOH336
AHOH517
ATRP81
APRO82
APHE83
AGLN85
APRO86
AVAL87
AASP88
ALYS91

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

222624

PDB entries from 2024-07-17

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