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7JJG

Crystal structure of the second bromodomain (BD2) of human TAF1 bound to ATR kinase inhibitor AZ20

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0005669cellular_componenttranscription factor TFIID complex
A0006366biological_processtranscription by RNA polymerase II
A0016251molecular_functionRNA polymerase II general transcription initiation factor activity
A0017025molecular_functionTBP-class protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue VCD A 1701
ChainResidue
ATRP1526
ATYR1601
ATHR1605
AEDO1702
AHOH1819
AHOH1843
APRO1527
AHIS1530
APRO1531
AVAL1532
AASN1533
APHE1536
AASN1583
ATYR1589

site_idAC2
Number of Residues6
Detailsbinding site for residue EDO A 1702
ChainResidue
AARG1565
AASP1608
AVCD1701
AHOH1807
AHOH1822
AHOH1830

site_idAC3
Number of Residues5
Detailsbinding site for residue GOL A 1703
ChainResidue
AASP1503
AALA1506
ALYS1534
AHIS1610
AGLU1627

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. SwpFhhpvNkkfvp..DYYkvIvnpMdletIrkniskhk..Yqsresflddvnl.IlaNSvkY
ChainResidueDetails
ASER1525-TYR1582

223532

PDB entries from 2024-08-07

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