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7ENE

Crystal structure of MERS-CoV 3CLpro in complex with the non-covalent inhibitor WU-04

Functional Information from GO Data
ChainGOidnamespacecontents
A0008233molecular_functionpeptidase activity
A0019082biological_processviral protein processing
B0008233molecular_functionpeptidase activity
B0019082biological_processviral protein processing
C0008233molecular_functionpeptidase activity
C0019082biological_processviral protein processing
D0008233molecular_functionpeptidase activity
D0019082biological_processviral protein processing
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue J7R A 401
ChainResidue
AHIS41
AGLU169
AASP190
ALYS191
AVAL193
BSER1
APHE143
ALEU144
ACYS145
AGLY146
ACYS148
AHIS166
AGLN167
AMET168

site_idAC2
Number of Residues16
Detailsbinding site for residue J7R B 401
ChainResidue
AHIS64
BHIS41
BLEU49
BPHE143
BLEU144
BCYS145
BGLY146
BCYS148
BHIS166
BGLN167
BGLU169
BASP190
BLYS191
BGLN192
BVAL193
BGLN195

site_idAC3
Number of Residues14
Detailsbinding site for residue J7R C 401
ChainResidue
CHIS41
CLEU49
CPHE143
CLEU144
CCYS145
CGLY146
CSER147
CCYS148
CHIS166
CGLN167
CGLU169
CLYS191
CGLN192
CVAL193

site_idAC4
Number of Residues15
Detailsbinding site for residue J7R D 401
ChainResidue
DHIS41
DPHE143
DLEU144
DCYS145
DGLY146
DSER147
DCYS148
DHIS166
DGLN167
DMET168
DGLU169
DASP190
DLYS191
DGLN192
DVAL193

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsActive site: {"description":"For 3CL-PRO activity","evidences":[{"source":"PROSITE-ProRule","id":"PRU00772","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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