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7CSI

Aminoglycoside 2'-N-acetyltransferase from Mycolicibacterium smegmatis-Complex with Coenzyme A and Sisomicin

Functional Information from GO Data
ChainGOidnamespacecontents
A0016746molecular_functionacyltransferase activity
A0016747molecular_functionacyltransferase activity, transferring groups other than amino-acyl groups
A0046677biological_processresponse to antibiotic
B0016746molecular_functionacyltransferase activity
B0016747molecular_functionacyltransferase activity, transferring groups other than amino-acyl groups
B0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue SIS A 301
ChainResidue
AASP54
ATRP210
ACOA302
AHOH416
AHOH448
AHOH474
AHOH508
AHOH527
AASP59
ASER141
AALA142
ASER143
AASP144
AGLU176
AASP177
AARG179

site_idAC2
Number of Residues21
Detailsbinding site for residue COA A 302
ChainResidue
APHE42
AVAL108
AALA109
AVAL110
AARG115
AGLY116
AASP117
AGLY118
ALEU119
AGLY120
ATHR121
AALA142
ASER143
ATYR150
ASIS301
AHOH414
AHOH439
AHOH450
AHOH457
AHOH543
BCOA302

site_idAC3
Number of Residues18
Detailsbinding site for residue SIS B 301
ChainResidue
BPHE42
BASP54
BASP59
BSER141
BALA142
BSER143
BASP144
BGLU176
BASP177
BTRP210
BCOA302
BHOH409
BHOH425
BHOH462
BHOH480
BHOH481
BHOH483
BHOH513

site_idAC4
Number of Residues26
Detailsbinding site for residue COA B 302
ChainResidue
ACOA302
BALA41
BPHE42
BVAL108
BALA109
BVAL110
BARG115
BGLY116
BASP117
BGLY118
BLEU119
BGLY120
BTHR121
BSER143
BILE145
BALA146
BPRO148
BMET149
BTYR150
BSIS301
BHOH403
BHOH406
BHOH407
BHOH418
BHOH426
BHOH451

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P9WQG9
ChainResidueDetails
AASP54
BARG115
BSER141
BGLU176
AGLU106
AVAL108
AARG115
ASER141
AGLU176
BASP54
BGLU106
BVAL108

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PDB entries from 2024-07-31

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