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7CS1

Aminoglycoside 2'-N-acetyltransferase from Mycolicibacterium smegmatis-Complex with Coenzyme A and Neomycin

Functional Information from GO Data
ChainGOidnamespacecontents
A0016746molecular_functionacyltransferase activity
A0016747molecular_functionacyltransferase activity, transferring groups other than amino-acyl groups
A0046677biological_processresponse to antibiotic
B0016746molecular_functionacyltransferase activity
B0016747molecular_functionacyltransferase activity, transferring groups other than amino-acyl groups
B0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues21
Detailsbinding site for residue NMY A 301
ChainResidue
APHE42
ASER143
AASP144
AARG147
AGLU176
AASP177
ATRP210
ACOA302
AHOH414
AHOH415
AHOH437
AASP44
AHOH458
AHOH495
AASP54
APHE55
AASP59
AGLU106
AALA107
ASER141
AALA142

site_idAC2
Number of Residues22
Detailsbinding site for residue COA A 302
ChainResidue
APHE42
AVAL108
AALA109
AVAL110
AARG115
AGLY116
AASP117
AGLY118
ALEU119
AGLY120
ATHR121
ASER143
AMET149
ANMY301
ACOA303
AHOH405
AHOH419
AHOH464
AHOH475
AHOH482
AHOH504
BCOA302

site_idAC3
Number of Residues10
Detailsbinding site for residue COA A 303
ChainResidue
AARG115
AGLY116
AALA152
ACOA302
AHOH475
BARG115
BGLY116
BASP117
BGLY118
BCOA302

site_idAC4
Number of Residues16
Detailsbinding site for residue NMY B 301
ChainResidue
BPHE42
BASP54
BPHE55
BASP59
BGLU106
BALA107
BSER141
BSER143
BGLU176
BASP177
BASP208
BTRP210
BCOA302
BHOH415
BHOH431
BHOH439

site_idAC5
Number of Residues21
Detailsbinding site for residue COA B 302
ChainResidue
ACOA302
ACOA303
BALA41
BPHE42
BVAL108
BALA109
BVAL110
BARG115
BGLY116
BASP117
BGLY118
BLEU119
BGLY120
BTHR121
BSER143
BPRO148
BMET149
BTYR150
BNMY301
BHOH410
BHOH441

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P9WQG9
ChainResidueDetails
AVAL108
AARG115
ASER141
AGLU176
BASP54
BGLU106
BVAL108
BARG115
BSER141
BGLU176
AGLU106
AASP54

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PDB entries from 2024-06-12

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