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7CJT

Crystal Structure of SETDB1 Tudor domain in complexed with (R,R)-59

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue G09 D 501
ChainResidue
DTHR210
DTHR212
DTYR268
DTRP275
DTYR277
DASP299
DTYR301
DGLU386

site_idAC2
Number of Residues11
Detailsbinding site for residue G09 A 501
ChainResidue
ATHR212
ATYR268
ATYR277
APHE297
AASP299
ATYR301
AGLU386
BASP270
BTRP275
BG09501
ATHR210

site_idAC3
Number of Residues6
Detailsbinding site for residue G09 B 501
ChainResidue
AG09501
BTHR212
BTYR268
BTRP275
BASP299
BGLU386

site_idAC4
Number of Residues15
Detailsbinding site for residue G09 C 501
ChainResidue
BASP331
BGLU334
BTHR338
BALA339
BPRO341
BASN342
CTHR210
CTHR212
CTYR268
CTRP275
CTYR277
CPHE297
CASP299
CTYR301
CGLU386

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues252
DetailsDomain: {"description":"Tudor 1"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues224
DetailsDomain: {"description":"Tudor 2"}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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