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7C9N

Crystal structure of SETDB1 tudor domain in complexed with Compound 1.

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue FN9 B 501
ChainResidue
ATRP275
AFN9501
BTHR212
BTYR268
BTRP275
BASP299
BTYR301
BGLU386

site_idAC2
Number of Residues7
Detailsbinding site for residue FN9 A 501
ChainResidue
AASP299
ATYR301
AGLU386
AARG394
BTRP275
BFN9501
ATYR268

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues126
DetailsDomain: {"description":"Tudor 1"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues112
DetailsDomain: {"description":"Tudor 2"}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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