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7C7V

Vitamin D3 receptor/lithochoric acid derivative complex

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue FKC A 501
ChainResidue
ATYR143
AVAL414
ALEU223
ASER271
ASER274
ATRP282
AHIS301
AILE306
AHIS393
ATYR397

site_idAC2
Number of Residues3
Detailsbinding site for residue FMT A 502
ChainResidue
ATHR276
AMET277
ALYS317

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues18
DetailsRegion: {"description":"Interaction with coactivator LXXLL motif","evidences":[{"source":"PubMed","id":"15065852","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"9aaTAD","evidences":[{"source":"UniProtKB","id":"P11473","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"15065852","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1RK3","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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