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7AXL

Crystal structure of the hPXR-LBD in complex with estradiol and heptachlor endo-epoxide

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue EST A 501
ChainResidue
AASP205
ALEU240
AMET243
ASER247
APHE251
AHIS407
AARG410
ALEU411

site_idAC2
Number of Residues8
Detailsbinding site for residue S65 A 502
ChainResidue
AMET243
AMET246
ASER247
AGLN285
APHE288
ATRP299
AHIS327
ALEU209

site_idAC3
Number of Residues6
Detailsbinding site for residue MPD A 503
ChainResidue
AHIS336
AGLU337
AGLU338
ALYS374
ATYR376
AGLU378

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
ASER247
AGLN285
AHIS407

224004

PDB entries from 2024-08-21

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