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7AXK

Crystal structure of the hPXR-LBD in complex with estradiol and endosulfan

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue EST A 501
ChainResidue
AASP205
ASER208
ASER247
APHE251
AHIS407
AARG410
ALEU411
AHOH745

site_idAC2
Number of Residues4
Detailsbinding site for residue MPD A 502
ChainResidue
AARG387
AHOH640
AHOH666
AGLU337

site_idAC3
Number of Residues11
Detailsbinding site for residue S68 A 503
ChainResidue
ALEU209
AMET243
ASER247
ACYS284
AGLN285
APHE288
ATRP299
ATYR306
AMET323
AHIS327
AHOH627

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"12578355","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1M13","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsModified residue: {"description":"Phosphothreonine; by PKC","evidences":[{"source":"PubMed","id":"26534988","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

249697

PDB entries from 2026-02-25

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