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7AXI

Crystal structure of the hPXR-LBD in complex with estradiol and cis-chlordane

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue EST A 501
ChainResidue
AASP205
AMET425
AS6E503
AS6H504
ASER208
ALEU240
AMET243
ASER247
APHE251
AHIS407
AARG410
ALEU411

site_idAC2
Number of Residues5
Detailsbinding site for residue MPD A 502
ChainResidue
AGLU337
ATYR340
AARG387
AHOH615
AHOH638

site_idAC3
Number of Residues9
Detailsbinding site for residue S6E A 503
ChainResidue
AMET243
ASER247
ACYS284
AGLN285
APHE288
ATRP299
AMET323
AEST501
AS6H504

site_idAC4
Number of Residues9
Detailsbinding site for residue S6H A 504
ChainResidue
AMET243
ASER247
ACYS284
AGLN285
APHE288
ATYR306
AMET323
AEST501
AS6E503

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
AHIS407
AGLN285
ASER247

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PDB entries from 2024-06-12

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