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7AXH

Crystal structure of the hPXR-LBD in complex with alpha-zearalanol

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue MPD A 502
ChainResidue
AGLU337
ATYR340
AARG387
AHOH616

site_idAC2
Number of Residues5
Detailsbinding site for residue IPA A 503
ChainResidue
ASER247
AGLN285
APHE288
AHIS407
A27J504

site_idAC3
Number of Residues11
Detailsbinding site for residue 27J A 504
ChainResidue
AVAL211
ALEU239
AHIS242
AMET243
AMET246
AGLN285
APHE288
ATRP299
ATYR306
AMET323
AIPA503

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
ASER247
AGLN285
AHIS407

224004

PDB entries from 2024-08-21

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