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7AXH

Crystal structure of the hPXR-LBD in complex with alpha-zearalanol

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue MPD A 502
ChainResidue
AGLU337
ATYR340
AARG387
AHOH616

site_idAC2
Number of Residues5
Detailsbinding site for residue IPA A 503
ChainResidue
ASER247
AGLN285
APHE288
AHIS407
A27J504

site_idAC3
Number of Residues11
Detailsbinding site for residue 27J A 504
ChainResidue
AVAL211
ALEU239
AHIS242
AMET243
AMET246
AGLN285
APHE288
ATRP299
ATYR306
AMET323
AIPA503

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"12578355","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1M13","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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