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7AXG

Crystal structure of the hPXR-LBD in complex with tributyltin

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue TBY A 501
ChainResidue
ACYS207
ATRP299
ATBY502

site_idAC2
Number of Residues8
Detailsbinding site for residue TBY A 502
ChainResidue
AHIS327
ATBY501
AMET243
AMET246
ASER247
APHE281
ACYS284
AGLN285

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
AHIS407
ASER247
AGLN285

219869

PDB entries from 2024-05-15

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