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7AXE

Crystal structure of the hPXR-LBD in complex with oxadiazon

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue GOL A 501
ChainResidue
ATHR290
ALEU335
AHIS336
AGLU337
AARG387
AHOH633
AHOH646
AHOH653

site_idAC2
Number of Residues11
Detailsbinding site for residue S6Z A 502
ChainResidue
AMET246
ASER247
ACYS284
AGLN285
APHE288
AMET323
AHIS407
ALEU411
APHE420
APHE429
AMET243

site_idAC3
Number of Residues5
Detailsbinding site for residue IPA A 503
ChainResidue
ATHR290
AVAL291
APHE292
AGLU300
ALYS331

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
ASER247
AGLN285
AHIS407

218853

PDB entries from 2024-04-24

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