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7AXA

Crystal structure of the hPXR-LBD in complex with clotrimazole

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue CL6 A 501
ChainResidue
ASER208
ALEU324
AHIS327
AHIS407
AHOH729
ALEU209
AVAL211
ASER247
AGLN285
APHE288
ATRP299
ATYR306
AMET323

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"12578355","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1M13","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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