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7AX9

Crystal structure of the hPXR-LBD in complex with cis-chlordane

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue S6H A 501
ChainResidue
ALEU209
AMET243
AMET246
ASER247
ACYS284
AGLN285
APHE288
ATRP299
AMET323

site_idAC2
Number of Residues2
Detailsbinding site for residue IPA A 502
ChainResidue
AGLU337
ATYR340

site_idAC3
Number of Residues1
Detailsbinding site for residue IPA A 503
ChainResidue
ALYS160

site_idAC4
Number of Residues1
Detailsbinding site for residue GOL A 505
ChainResidue
AHIS407

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"12578355","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1M13","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

244349

PDB entries from 2025-11-05

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