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7AWX

Structure of the FKBP51FK1 domain in complex with the macrocyclic SAFit analogue 55

Functional Information from GO Data
ChainGOidnamespacecontents
A0003755molecular_functionpeptidyl-prolyl cis-trans isomerase activity
B0003755molecular_functionpeptidyl-prolyl cis-trans isomerase activity
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue S5W A 201
ChainResidue
ATYR57
ASER118
APHE130
BGLN85
BS5W201
AGLY59
AASP68
APHE77
AGLN85
AVAL86
AILE87
ATRP90
ATYR113

site_idAC2
Number of Residues16
Detailsbinding site for residue S5W B 201
ChainResidue
ALEU119
AS5W201
BTYR57
BGLY59
BASP68
BPHE77
BGLY84
BGLN85
BVAL86
BILE87
BTRP90
BALA112
BTYR113
BSER118
BILE122
BPHE130

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: N6-acetyllysine => ECO:0000269|PubMed:28147277
ChainResidueDetails
ALYS28
BLYS28

223790

PDB entries from 2024-08-14

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