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7AOU

The Fk1 domain of FKBP51 in complex with (2'R,5'S,12'R)-12'-cyclohexyl-2'-[2-(3,4-dimethoxyphenyl)ethyl]-3',19'-dioxa-10',13',16'-triazaspiro[cyclopropane-1,15'- tricyclo[18.3.1.0-5,10]tetracosane]-1'(24'),20',22'-triene-4',11',14',17'-tetrone

Functional Information from GO Data
ChainGOidnamespacecontents
A0003755molecular_functionpeptidyl-prolyl cis-trans isomerase activity
Functional Information from PDB Data
site_idAC1
Number of Residues20
Detailsbinding site for residue RTT A 301
ChainResidue
ALYS28
AVAL86
AILE87
ATRP90
AALA112
ATYR113
ALYS121
AHOH431
AHOH484
AHOH485
AHOH514
ALYS29
AHOH526
AASP30
AARG31
ATYR57
ASER70
APHE77
AGLY84
AGLN85

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0000269|PubMed:28147277
ChainResidueDetails
ALYS28

221051

PDB entries from 2024-06-12

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