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7AMD

In situ assembly of choline acetyltransferase ligands by a hydrothiolation reaction reveals key determinants for inhibitor design

Functional Information from GO Data
ChainGOidnamespacecontents
A0016746molecular_functionacyltransferase activity
Functional Information from PROSITE/UniProt
site_idPS00439
Number of Residues16
DetailsACYLTRANSF_C_1 Acyltransferases ChoActase / COT / CPT family signature 1. LPkLPVPpLqQTLatY
ChainResidueDetails
ALEU13-TYR28

site_idPS00440
Number of Residues28
DetailsACYLTRANSF_C_2 Acyltransferases ChoActase / COT / CPT family signature 2. RWyDKsLqFVvgrDGtcgvvcEHspfDG
ChainResidueDetails
AARG302-GLY329

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsActive site: {"description":"Proton acceptor"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues14
DetailsBinding site: {}
ChainResidueDetails

239149

PDB entries from 2025-07-23

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