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7A1C

LdtMT2 with covalent adduct derived from N-Thio-beta-lactam 1a

Functional Information from GO Data
ChainGOidnamespacecontents
A0016740molecular_functiontransferase activity
B0016740molecular_functiontransferase activity
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: Proton donor/acceptor => ECO:0000255|PROSITE-ProRule:PRU01373, ECO:0000305|PubMed:23519417
ChainResidueDetails
AHIS336
BHIS336

site_idSWS_FT_FI2
Number of Residues2
DetailsACT_SITE: Nucleophile => ECO:0000255|PROSITE-ProRule:PRU01373, ECO:0000269|PubMed:23519417
ChainResidueDetails
ASCH354
BSCH354

site_idSWS_FT_FI3
Number of Residues6
DetailsBINDING:
ChainResidueDetails
AASP232
AGLU235
AGLY236
BASP232
BGLU235
BGLY236

site_idSWS_FT_FI4
Number of Residues6
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
ATYR318
ASER331
AASN356
BTYR318
BSER331
BASN356

site_idSWS_FT_FI5
Number of Residues2
DetailsSITE: Binds to carbapenem drug (covalent)
ChainResidueDetails
ASCH354
BSCH354

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PDB entries from 2024-07-10

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