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6ZC7

Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling

Functional Information from GO Data
ChainGOidnamespacecontents
A0016055biological_processWnt signaling pathway
B0016055biological_processWnt signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue V31 A 401
ChainResidue
APHE259
AV31402
BILE305
ALEU260
AGLY261
AILE262
AVAL316
ALEU319
AARG320
AVAL323
AHIS324

site_idAC2
Number of Residues10
Detailsbinding site for residue V31 A 402
ChainResidue
AILE262
ASER263
ASER280
AMET282
AV31401
BASN303
BGLU304
BILE305
BHOH605
BHOH612

site_idAC3
Number of Residues9
Detailsbinding site for residue V31 B 401
ChainResidue
BPHE259
BLEU260
BGLY261
BILE262
BMET282
BARG320
BVAL323
BHIS324
BHOH516

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Symmetric dimethylarginine; by PRMT7; alternate => ECO:0000269|PubMed:23150776
ChainResidueDetails
AARG271
BARG271

237992

PDB entries from 2025-06-25

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