Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 25 |
Details | binding site for residue A1R A 401 |
Chain | Residue |
A | ASP226 |
A | LEU330 |
A | SER332 |
A | ALA333 |
A | GLY334 |
A | ILE335 |
A | PHE336 |
A | ALA358 |
A | PHE360 |
A | A1R406 |
A | HOH520 |
A | ILE227 |
A | HOH521 |
A | HOH540 |
A | HOH547 |
A | HOH576 |
A | HOH578 |
A | HOH583 |
A | ALA242 |
A | ASN244 |
A | LYS248 |
A | GLY250 |
A | GLY251 |
A | VAL253 |
A | ALA254 |
site_id | AC2 |
Number of Residues | 5 |
Details | binding site for residue EDO A 402 |
Chain | Residue |
A | LEU279 |
A | LYS280 |
A | GLY283 |
A | SER284 |
A | HOH580 |
site_id | AC3 |
Number of Residues | 7 |
Details | binding site for residue EDO A 403 |
Chain | Residue |
A | GLY212 |
A | LYS223 |
A | ASN224 |
A | TYR365 |
A | HOH555 |
A | HOH560 |
A | HOH563 |
site_id | AC4 |
Number of Residues | 9 |
Details | binding site for residue GOL A 404 |
Chain | Residue |
A | ASN244 |
A | VAL245 |
A | VAL281 |
A | VAL300 |
A | GLY301 |
A | ASN303 |
A | LYS306 |
A | GLU308 |
A | PHE336 |
site_id | AC5 |
Number of Residues | 5 |
Details | binding site for residue EDO A 405 |
Chain | Residue |
A | GLU318 |
A | ASP349 |
A | THR350 |
A | HOH513 |
B | MPO403 |
site_id | AC6 |
Number of Residues | 12 |
Details | binding site for residue A1R A 406 |
Chain | Residue |
A | ASP226 |
A | ILE335 |
A | PHE360 |
A | A1R401 |
A | HOH504 |
A | HOH516 |
A | HOH517 |
A | HOH528 |
B | ASN321 |
B | GLU324 |
B | ARG352 |
B | HOH505 |
site_id | AC7 |
Number of Residues | 3 |
Details | binding site for residue NA A 407 |
Chain | Residue |
A | ASN363 |
A | ASP366 |
A | HOH603 |
site_id | AC8 |
Number of Residues | 2 |
Details | binding site for residue NA A 408 |
Chain | Residue |
A | ASP339 |
A | ILE341 |
site_id | AC9 |
Number of Residues | 30 |
Details | binding site for residue A1R B 401 |
Chain | Residue |
B | ASP226 |
B | ILE227 |
B | ALA242 |
B | ASN244 |
B | LYS248 |
B | GLY250 |
B | GLY251 |
B | GLY252 |
B | VAL253 |
B | ALA254 |
B | LEU330 |
B | SER332 |
B | ALA333 |
B | GLY334 |
B | ILE335 |
B | PHE336 |
B | ALA358 |
B | PHE360 |
B | MPO403 |
B | HOH502 |
B | HOH517 |
B | HOH522 |
B | HOH526 |
B | HOH530 |
B | HOH531 |
B | HOH539 |
B | HOH541 |
B | HOH567 |
B | HOH572 |
B | HOH576 |
site_id | AD1 |
Number of Residues | 3 |
Details | binding site for residue GOL B 402 |
Chain | Residue |
B | GLY251 |
B | HOH517 |
B | GLY250 |
site_id | AD2 |
Number of Residues | 11 |
Details | binding site for residue MPO B 403 |
Chain | Residue |
A | ASN321 |
A | ARG352 |
A | THR353 |
A | EDO405 |
A | HOH552 |
B | ASP226 |
B | GLU229 |
B | PHE360 |
B | A1R401 |
B | HOH530 |
B | HOH571 |
site_id | AD3 |
Number of Residues | 3 |
Details | binding site for residue EDO B 404 |
Chain | Residue |
B | ASN276 |
B | HOH507 |
B | HOH590 |
site_id | AD4 |
Number of Residues | 4 |
Details | binding site for residue NA B 405 |
Chain | Residue |
B | ASN263 |
B | GLN266 |
B | HOH570 |
B | HOH622 |
site_id | AD5 |
Number of Residues | 26 |
Details | binding site for residue A1R C 401 |
Chain | Residue |
C | ASP226 |
C | ILE227 |
C | ALA242 |
C | ASN244 |
C | LYS248 |
C | GLY250 |
C | GLY251 |
C | VAL253 |
C | ALA254 |
C | LEU330 |
C | SER332 |
C | ALA333 |
C | GLY334 |
C | ILE335 |
C | PHE336 |
C | ALA358 |
C | PHE360 |
C | HOH551 |
C | HOH559 |
C | HOH560 |
C | HOH569 |
C | HOH573 |
C | HOH578 |
C | HOH590 |
C | HOH592 |
C | HOH613 |
site_id | AD6 |
Number of Residues | 9 |
Details | binding site for residue GOL C 402 |
Chain | Residue |
C | THR217 |
C | ASP218 |
C | ASN219 |
C | VAL348 |
C | GOL406 |
C | HOH502 |
C | HOH513 |
C | HOH577 |
C | HOH587 |
site_id | AD7 |
Number of Residues | 7 |
Details | binding site for residue EDO C 403 |
Chain | Residue |
C | HIS249 |
C | GLY250 |
C | GLY255 |
C | ASN258 |
C | LYS259 |
C | HOH516 |
C | HOH616 |
site_id | AD8 |
Number of Residues | 4 |
Details | binding site for residue EDO C 404 |
Chain | Residue |
C | TYR221 |
C | ASN354 |
C | HOH523 |
C | HOH524 |
site_id | AD9 |
Number of Residues | 7 |
Details | binding site for residue EDO C 405 |
Chain | Residue |
C | PHE210 |
C | SER211 |
C | GLY212 |
C | TYR213 |
C | TYR356 |
C | HOH526 |
C | HOH593 |
site_id | AE1 |
Number of Residues | 7 |
Details | binding site for residue GOL C 406 |
Chain | Residue |
C | ASN219 |
C | VAL348 |
C | ASP349 |
C | THR350 |
C | VAL351 |
C | ARG352 |
C | GOL402 |
site_id | AE2 |
Number of Residues | 18 |
Details | binding site for residue A1R C 407 |
Chain | Residue |
C | ASN321 |
C | GLU324 |
C | ARG352 |
C | THR353 |
C | HOH518 |
C | HOH547 |
C | HOH553 |
C | HOH582 |
C | HOH604 |
D | ASP226 |
D | GLU229 |
D | GLY252 |
D | GLY334 |
D | PHE360 |
D | A1R401 |
D | EDO408 |
D | HOH533 |
D | HOH538 |
site_id | AE3 |
Number of Residues | 1 |
Details | binding site for residue NA C 408 |
site_id | AE4 |
Number of Residues | 2 |
Details | binding site for residue NA C 409 |
Chain | Residue |
C | LEU279 |
C | LYS280 |
site_id | AE5 |
Number of Residues | 3 |
Details | binding site for residue NA C 410 |
Chain | Residue |
C | HIS342 |
C | ARG345 |
C | HOH528 |
site_id | AE6 |
Number of Residues | 3 |
Details | binding site for residue NA C 411 |
Chain | Residue |
C | GLY251 |
C | ILE335 |
C | HOH714 |
site_id | AE7 |
Number of Residues | 25 |
Details | binding site for residue A1R D 401 |
Chain | Residue |
C | A1R407 |
D | ASP226 |
D | ILE227 |
D | ALA242 |
D | ASN244 |
D | LYS248 |
D | GLY250 |
D | GLY251 |
D | VAL253 |
D | ALA254 |
D | LEU330 |
D | SER332 |
D | ALA333 |
D | GLY334 |
D | ILE335 |
D | PHE336 |
D | ALA358 |
D | PHE360 |
D | EDO404 |
D | HOH520 |
D | HOH531 |
D | HOH533 |
D | HOH546 |
D | HOH557 |
D | HOH602 |
site_id | AE8 |
Number of Residues | 7 |
Details | binding site for residue GOL D 402 |
Chain | Residue |
D | VAL286 |
D | LEU287 |
D | SER288 |
D | LYS294 |
D | HIS295 |
D | HOH522 |
D | HOH529 |
site_id | AE9 |
Number of Residues | 4 |
Details | binding site for residue EDO D 403 |
Chain | Residue |
D | HIS249 |
D | GLN266 |
D | HOH511 |
D | HOH575 |
site_id | AF1 |
Number of Residues | 6 |
Details | binding site for residue EDO D 404 |
Chain | Residue |
D | ASN244 |
D | LYS248 |
D | GLY250 |
D | ILE335 |
D | A1R401 |
D | NA410 |
site_id | AF2 |
Number of Residues | 7 |
Details | binding site for residue EDO D 405 |
Chain | Residue |
C | LYS362 |
D | VAL286 |
D | ASN319 |
D | GLN322 |
D | HIS323 |
D | HOH571 |
D | HOH576 |
site_id | AF3 |
Number of Residues | 5 |
Details | binding site for residue EDO D 406 |
Chain | Residue |
C | GLU229 |
C | HOH609 |
D | ASN321 |
D | ARG352 |
D | HOH508 |
site_id | AF4 |
Number of Residues | 3 |
Details | binding site for residue EDO D 407 |
Chain | Residue |
D | PRO340 |
D | HOH515 |
D | HOH516 |
site_id | AF5 |
Number of Residues | 1 |
Details | binding site for residue EDO D 408 |
site_id | AF6 |
Number of Residues | 2 |
Details | binding site for residue NA D 409 |
Chain | Residue |
D | THR237 |
D | VAL325 |
site_id | AF7 |
Number of Residues | 2 |
Details | binding site for residue NA D 410 |
Chain | Residue |
D | EDO404 |
D | HOH510 |