6Y7K
Structure of the BRD9 bromodomain and compound 27
Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 8 |
| Details | binding site for residue OEZ A 700 |
| Chain | Residue |
| A | PHE160 |
| A | PHE161 |
| A | PHE163 |
| A | ILE169 |
| A | ASN216 |
| A | TYR222 |
| A | HOH815 |
| A | HOH896 |
| site_id | AC2 |
| Number of Residues | 4 |
| Details | binding site for residue EDO A 701 |
| Chain | Residue |
| A | GLY233 |
| A | HOH842 |
| A | HOH874 |
| A | LYS206 |
| site_id | AC3 |
| Number of Residues | 5 |
| Details | binding site for residue EDO A 702 |
| Chain | Residue |
| A | LYS189 |
| A | HIS231 |
| A | LYS235 |
| A | HOH818 |
| A | HOH823 |
| site_id | AC4 |
| Number of Residues | 5 |
| Details | binding site for residue NA A 703 |
| Chain | Residue |
| A | LYS178 |
| A | HIS179 |
| A | ASN211 |
| A | HOH889 |
| A | HOH939 |
| site_id | AC5 |
| Number of Residues | 4 |
| Details | binding site for residue NA A 704 |
| Chain | Residue |
| A | HIS147 |
| A | MET236 |
| A | ARG241 |
| A | HOH907 |
Functional Information from SwissProt/UniProt
| site_id | SWS_FT_FI1 |
| Number of Residues | 2 |
| Details | Region: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]} |
| Chain | Residue | Details |
| site_id | SWS_FT_FI2 |
| Number of Residues | 2 |
| Details | Site: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]} |
| Chain | Residue | Details |






