6Y7J
Structure of the BRD9 bromodomain and compound 15
Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 10 |
| Details | binding site for residue OF5 A 700 |
| Chain | Residue |
| A | PHE160 |
| B | HIS158 |
| A | PHE163 |
| A | VAL165 |
| A | ILE169 |
| A | ASN216 |
| A | TYR222 |
| A | HOH821 |
| A | HOH841 |
| A | HOH866 |
| site_id | AC2 |
| Number of Residues | 10 |
| Details | binding site for residue OF5 B 700 |
| Chain | Residue |
| A | HIS158 |
| A | PHE160 |
| B | PHE160 |
| B | PHE163 |
| B | VAL165 |
| B | ILE169 |
| B | ASN216 |
| B | TYR222 |
| B | HOH804 |
| B | HOH870 |
| site_id | AC3 |
| Number of Residues | 4 |
| Details | binding site for residue ACT B 701 |
| Chain | Residue |
| B | ILE176 |
| B | ILE177 |
| B | LYS178 |
| B | HOH846 |
| site_id | AC4 |
| Number of Residues | 2 |
| Details | binding site for residue CL B 702 |
| Chain | Residue |
| B | GLY172 |
| B | HOH867 |
Functional Information from SwissProt/UniProt
| site_id | SWS_FT_FI1 |
| Number of Residues | 4 |
| Details | Region: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]} |
| Chain | Residue | Details |
| site_id | SWS_FT_FI2 |
| Number of Residues | 4 |
| Details | Site: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]} |
| Chain | Residue | Details |






