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6XZI

Structure of zVDR LBD-calcitriol in complex with chimera 11

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue VDX A 501
ChainResidue
ATYR175
AHIS423
ASER265
AARG302
ASER303
ASER306
ATRP314
ACYS316
AVAL328
AHIS333

site_idAC2
Number of Residues7
Detailsbinding site for residue ACT A 502
ChainResidue
ATHR174
ATYR175
AASP176
ATYR264
ALYS268
AARG302
AHOH638

site_idAC3
Number of Residues5
Detailsbinding site for residues URL A 502 and UIL B 701
ChainResidue
ALYS274
AARG280
BILE689
BLEU690
BOUK691

site_idAC4
Number of Residues8
Detailsbinding site for residues UIL B 701 and OUK B 691
ChainResidue
ALYS274
AGLU285
AILE288
BURL693
BHIS687
BLYS688
BILE689
BLEU690

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:17218092, ECO:0007744|PDB:2HC4
ChainResidueDetails
ATYR175
ASER265
AARG302
ASER306
AHIS333
AHIS423

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PDB entries from 2024-07-17

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