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6XV7

CRYSTAL STRUCTURE OF BRD4-BD1 WITH COMPOUND 2

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 201
ChainResidue
ATYR65
ATYR137
AGLU151
ALYS160
AHOH301
AHOH324

site_idAC2
Number of Residues6
Detailsbinding site for residue EDO A 202
ChainResidue
ATHR103
AASN135
AHOH361
AILE100
AILE101
ALYS102

site_idAC3
Number of Residues6
Detailsbinding site for residue EDO A 203
ChainResidue
APRO46
APRO47
APRO48
APRO104
ATRP120
AHOH318

site_idAC4
Number of Residues11
Detailsbinding site for residue O2Q A 204
ChainResidue
ATRP81
APRO82
AVAL87
ALEU92
AASP96
ALYS99
AASN140
AASP145
AILE146
AMET149
AHOH313

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues106
DetailsDomain: {"description":"Bromo 1","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

247947

PDB entries from 2026-01-21

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