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6XFV

CRYSTAL STRUCTURE OF RAR-RELATED ORPHAN RECEPTOR C IN COMPLEX WITH A NOVEL INVERSE AGONIST

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue V27 A 500
ChainResidue
ALEU266
ALEU375
AILE379
AHIS458
AARG461
ALEU462
AHOH605
AHOH630
ACYS299
AHIS302
AVAL340
AMET344
APHE357
AGLU358
APHE367
ALEU370

site_idAC2
Number of Residues13
Detailsbinding site for residue V27 B 500
ChainResidue
BLEU266
BCYS299
BALA300
BHIS302
BVAL340
BMET344
BPHE357
BGLU358
BPHE367
BLEU370
BHIS458
BARG461
BLEU462

222415

PDB entries from 2024-07-10

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