6XFV
CRYSTAL STRUCTURE OF RAR-RELATED ORPHAN RECEPTOR C IN COMPLEX WITH A NOVEL INVERSE AGONIST
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0003677 | molecular_function | DNA binding |
A | 0004879 | molecular_function | nuclear receptor activity |
A | 0005634 | cellular_component | nucleus |
A | 0006355 | biological_process | regulation of DNA-templated transcription |
B | 0003677 | molecular_function | DNA binding |
B | 0004879 | molecular_function | nuclear receptor activity |
B | 0005634 | cellular_component | nucleus |
B | 0006355 | biological_process | regulation of DNA-templated transcription |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 16 |
Details | binding site for residue V27 A 500 |
Chain | Residue |
A | LEU266 |
A | LEU375 |
A | ILE379 |
A | HIS458 |
A | ARG461 |
A | LEU462 |
A | HOH605 |
A | HOH630 |
A | CYS299 |
A | HIS302 |
A | VAL340 |
A | MET344 |
A | PHE357 |
A | GLU358 |
A | PHE367 |
A | LEU370 |
site_id | AC2 |
Number of Residues | 13 |
Details | binding site for residue V27 B 500 |
Chain | Residue |
B | LEU266 |
B | CYS299 |
B | ALA300 |
B | HIS302 |
B | VAL340 |
B | MET344 |
B | PHE357 |
B | GLU358 |
B | PHE367 |
B | LEU370 |
B | HIS458 |
B | ARG461 |
B | LEU462 |