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6WE7

HIV Integrase core domain in complex with inhibitor 3-methyl-2-{5-methyl-2-[2-(thiophen-2-yl)ethynyl]-1- benzofuran-3-yl}butanoic acid

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue SO4 A 301
ChainResidue
ASER123
ATHR124
ATHR125

site_idAC2
Number of Residues4
Detailsbinding site for residue SO4 A 302
ChainResidue
ACSD65
ATHR66
AHIS67
ATYR194

site_idAC3
Number of Residues5
Detailsbinding site for residue SO4 A 303
ChainResidue
AGLN137
ALYS185
AARG187
APHE121
ALYS127

site_idAC4
Number of Residues8
Detailsbinding site for residue SO4 A 304
ChainResidue
ASER81
AGLY82
AHIS183
ALYS188
AARG199
AHOH402
AHOH410
AHOH419

site_idAC5
Number of Residues5
Detailsbinding site for residue SO4 A 305
ChainResidue
ASER57
APRO58
AGLY59
AILE60
ALYS111

site_idAC6
Number of Residues2
Detailsbinding site for residue IOD A 306
ChainResidue
AGLY70
AARG199

site_idAC7
Number of Residues2
Detailsbinding site for residue IOD A 307
ChainResidue
ALYS71
ALYS173

site_idAC8
Number of Residues11
Detailsbinding site for residue TXM A 308
ChainResidue
AGLN95
AGLU96
AALA98
ATYR99
ALEU102
AALA129
AALA169
AGLU170
AHIS171
ATHR174
AMET178

219869

PDB entries from 2024-05-15

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