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6W42

HIV Integrase core domain in complex with inhibitor 2-(5-methyl-2-(2-(thiophen-2-yl)ethynyl)-1-benzofuran-3-yl)acetic acid

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue SO4 A 301
ChainResidue
AGLY94
ALYS111
ASER123
ATHR124
ATHR125

site_idAC2
Number of Residues2
Detailsbinding site for residue SO4 A 302
ChainResidue
ATHR66
AHIS67

site_idAC3
Number of Residues1
Detailsbinding site for residue IOD A 304
ChainResidue
AGLY70

site_idAC4
Number of Residues1
Detailsbinding site for residue IOD A 305
ChainResidue
AGLN137

site_idAC5
Number of Residues1
Detailsbinding site for residue IOD A 306
ChainResidue
ALYS173

site_idAC6
Number of Residues14
Detailsbinding site for residue SJY A 307
ChainResidue
AGLN95
AGLU96
AALA98
ATYR99
ALEU102
ATHR125
AALA128
AALA129
AALA169
AGLU170
AHIS171
ALYS173
ATHR174
AMET178

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING:
ChainResidueDetails
AASP64
AASP116

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P04585
ChainResidueDetails
AGLU152

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PDB entries from 2024-07-24

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