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6W0U

HIV Integrase core domain in complex with inhibitor 2-(2-ethynyl-5-methyl-1-benzofuran-3-yl)acetic acid

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue S0Y A 301
ChainResidue
AGLN95
AMET178
ATYR99
ALEU102
ATHR125
AALA129
AALA169
AGLU170
AHIS171
ATHR174

site_idAC2
Number of Residues5
Detailsbinding site for residue SO4 A 302
ChainResidue
ATHR66
AHIS67
AASN155
ALYS159
ATYR194

site_idAC3
Number of Residues1
Detailsbinding site for residue IOD A 303
ChainResidue
AGLN137

site_idAC4
Number of Residues2
Detailsbinding site for residue IOD A 304
ChainResidue
AHIS67
AGLY70

site_idAC5
Number of Residues2
Detailsbinding site for residue IOD A 305
ChainResidue
ALYS173
AHOH426

site_idAC6
Number of Residues3
Detailsbinding site for residue IOD A 306
ChainResidue
ASER123
ATHR124
ATHR125

site_idAC7
Number of Residues1
Detailsbinding site for residue IOD A 307
ChainResidue
APRO142

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI2
Number of Residues2
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues1
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"P04585","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

247947

PDB entries from 2026-01-21

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