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6VIZ

BRD4_Bromodomain1 complex with pyrrolopyridone compound 27

Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue QYY A 201
ChainResidue
ATRP81
AHOH306
AHOH313
CTRP81
CQYY201
APRO82
AGLN85
AVAL87
AASP88
ALEU92
AASN140
ALYS141
AILE146

site_idAC2
Number of Residues15
Detailsbinding site for residue QYY B 201
ChainResidue
BTRP81
BTRP81
BPRO82
BPHE83
BGLN85
BVAL87
BASP88
BLYS91
BLEU92
BLEU94
BASN140
BLYS141
BILE146
BHOH303
BHOH304

site_idAC3
Number of Residues14
Detailsbinding site for residue QYY C 201
ChainResidue
ATRP81
AQYY201
CTRP81
CPRO82
CPHE83
CGLN85
CVAL87
CASP88
CLYS91
CLEU92
CLEU94
CASN140
CILE146
CHOH303

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140
BASN140
CASN140

site_idSWS_FT_FI2
Number of Residues6
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99
BLYS99
CLYS99

222624

PDB entries from 2024-07-17

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